SCHEMBL4007142

SCHEMBL4007142

COc1ncnc2c1c(Br)cn2CC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FLT4 P35916 1/20 0.43
KDR P35968 1/20 0.43
CSNK2A1 P68400 2/20 0.38
CSNK2A2 P19784 1/20 0.38
HSD17B10 Q99714 1/20 0.37
CCR4 P51679 1/20 0.36
PTGS2 P35354 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
KLKB1 P03952 1/20 0.34
HPGD P15428 1/20 0.32
ALDH1A1 P00352 2/20 0.32
ADORA2B P29275 1/20 0.32
SRC P12931 1/20 0.32
HIPK2 Q9H2X6 1/20 0.32
KDM4E B2RXH2 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
EPHX2 P34913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4008751 0.80 CSNK2A2 (0.35) KDRCSNK2A1CSNK2A2ALDH1A1ADORA2B
SCHEMBL23885536 0.79 ADK (0.43) KDRALDH1A1ADORA2BSRC
SCHEMBL4005517 0.79 ADK (0.42) CSNK2A1CSNK2A2HDAC6SRCEPHX2
SCHEMBL4008754 0.76 FLT4 (0.44) FLT4KDRCCR4HPGDALDH1A1
SCHEMBL4007971 0.75 PTGS2 (0.48) HSD17B10PTGS2ALDH1A1SRCKDM4E
SCHEMBL4014223 0.74 HTT (0.42) HPGDALDH1A1KDM4EPOLBMAPT
SCHEMBL8769186 0.73 FLT4 (0.72) FLT4KDRCSNK2A1CSNK2A2PTGS2
SCHEMBL2236505 0.73 DGAT1 (0.38)
SCHEMBL4005527 0.72 MAPT (0.44) CSNK2A1MAPT
SCHEMBL4008412 0.69 CSNK2A2 (0.38) CSNK2A1CSNK2A2PTGS2HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed