SCHEMBL4012449

SCHEMBL4012449

CCOC(=O)Cc1ccc[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
HSD17B10 Q99714 2/20 0.48
CHEK1 O14757 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 2/20 0.42
KMT2A Q03164 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
GAA P10253 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
RECQL P46063 1/20 0.40
TSHR P16473 2/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4018484 1.00 PKM (0.49) PKMSMN1; SMN2HSD17B10CHEK1ALDH1A1
SCHEMBL1078882 0.83 CYP4F2 (0.51) PKMSMN1; SMN2HSD17B10ALDH1A1LMNA
SCHEMBL4802900 0.81 TSHR (0.45) SMN1; SMN2HSD17B10ALDH1A1LMNAKMT2A
SCHEMBL10813508 0.81 TSHR (0.36) SMN1; SMN2HSD17B10ALDH1A1KMT2ATDP1
SCHEMBL10511460 0.81 ALDH1A1 (0.40) PKMSMN1; SMN2HSD17B10ALDH1A1LMNA
SCHEMBL29225340 0.78 ALDH1A1 (0.64) ALDH1A1LMNAKMT2ATDP1L3MBTL1
SCHEMBL16111244 0.78 KMT2A (0.52) PKMSMN1; SMN2HSD17B10ALDH1A1LMNA
SCHEMBL7963890 0.78 CYP3A4 (0.45) PKMSMN1; SMN2HSD17B10ALDH1A1LMNA
SCHEMBL23500951 0.77 RAB9A (0.49) SMN1; SMN2ALDH1A1KMT2AKDM4EMEN1
SCHEMBL10362177 0.76 MAOA (0.36) KMT2ATDP1GAAL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10442874-B2 Heterocyclic organic compounds as electron donors for polyolefin catalysts FORMOSA PLASTICS CORPORATION, U.S.A. (US) 2019-10-15 US disclosed
US-9951152-B2 Heterocyclic organic compounds as electron donors for polyolefin catalysts FORMOSA PLASTICS CORPORATION, U.S.A. (US) 2018-04-24 US disclosed
US-20140058053-A1 Heterocyclic Organic Compounds As Electron Donors for Polyolefin Catalysts FORMOSA PLASTICS CORPORATION USA (US) 2014-02-27 US disclosed
US-8575283-B1 Heterocyclic organic compounds as electron donors for polyolefin catalysts FORMOSA PLASTICS CORPORATION, U.S.A. (US) 2013-11-05 US disclosed
WO-2009015180-A2 NOVEL COMPOUNDS AND METHODS OF USING THEM SYNDAX PHARMACEUTICALS, INC. (US) 2009-01-29 WO disclosed
US-7326788-B2 Selective, potent small molecule protein tyrosine kinase inhibitors; such as 6-chloro-3-(3-methyl-isoxazol-5-yl)-4-(pyridin-4-yl)-1H-quinolin-2-one JANSSEN PHARMACEUTICA N.V. (BE) 2008-02-05 US disclosed
EP-1660087-A2 QUINOLINONE DERIVATIVES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2006-05-31 EP disclosed
US-20050049274-A1 Quinolinone derivatives as inhibitors of c-fms kinase JANSSEN PHARMACEUTICA, N.V. (BE) 2005-03-03 US disclosed
WO-2005009967-A2 QUINOLINONE DERIVATIVES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA, N.V. (BE) 2005-02-03 WO disclosed
CN-1066726-C Pyrrole derivatives HOFFMANN LA ROCHE (CH) 2001-06-06 CN disclosed
CN-1132206-A Pyrrole derivatives HOFFMANN LA ROCHE (CH) 1996-10-02 CN disclosed
US-4136097-A COPPER(II) COMPLEX AS PROMOTER MCNEIL LABORATORIES, INC. (US) 1979-01-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050049274-A1 Quinolinone derivatives as inhibitors of c-fms kinase FLT3, ABL1, FES PKM 1156/4885SMN1; SMN2 4293/4885HSD17B10 4321/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.