SCHEMBL4018620

SCHEMBL4018620

COC(=O)N(N)c1ccccc1C#N

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 4/20 0.40
TSHR P16473 3/20 0.40
HPGD P15428 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
TDP1 Q9NUW8 1/20 0.38
MAPK1 P28482 1/20 0.38
KDM4E B2RXH2 2/20 0.37
TP53 P04637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
POLB P06746 1/20 0.37
LMNA P02545 1/20 0.36
KMT2A Q03164 1/20 0.36
NLRP3 Q96P20 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8544711 0.82 GAA (0.44) GAASMN1; SMN2ALDH1A1TSHRHPGD
SCHEMBL26631742 0.72 ALDH1A1 (0.47) GAASMN1; SMN2ALDH1A1TSHRHPGD
SCHEMBL514812 0.71 ALDH1A1 (0.39) GAASMN1; SMN2ALDH1A1TSHRHPGD
SCHEMBL9631333 0.70 ALDH1A1 (0.48) SMN1; SMN2ALDH1A1TSHRHPGDRAB9A
SCHEMBL11800729 0.70 GAA (0.40) GAASMN1; SMN2ALDH1A1TSHRHPGD
SCHEMBL4107497 0.70 L3MBTL1 (0.47) ALDH1A1TSHRHPGDL3MBTL1TDP1
SCHEMBL27701441 0.69 POLB (0.42) GAASMN1; SMN2ALDH1A1TSHRL3MBTL1
SCHEMBL17086067 0.69 ALDH1A1 (0.41) GAASMN1; SMN2ALDH1A1TSHRNPC1
SCHEMBL8835734 0.69 ALDH1A1 (0.49) GAAALDH1A1TSHRL3MBTL1NPC1
SCHEMBL8983982 0.69 PDK1 (0.40) GAASMN1; SMN2ALDH1A1TSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009089042-A1 PYRAZOLE PYRAZINE AMINE COMPOUNDS AS KINASE INHIBITORS, COMPOSITIONS THEREOF AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, LLC (US) 2009-07-16 WO disclosed