SCHEMBL4019325

SCHEMBL4019325

COCCn1c(-c2c[nH]nc2Cc2cccc(C(F)(F)F)c2)nc2[nH]c(=O)[nH]c(=O)c21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.42
HTT P42858 1/20 0.42
KDM4E B2RXH2 3/20 0.37
ALDH1A1 P00352 3/20 0.37
HSD17B10 Q99714 1/20 0.37
CNR2 P34972 2/20 0.37
RECQL P46063 2/20 0.36
GAA P10253 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
PARP1 P09874 2/20 0.36
NR3C1 P04150 1/20 0.35
GPR52 Q9Y2T5 1/20 0.35
TPH1 P17752 1/20 0.35
TPH2 Q8IWU9 1/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
PKM P14618 1/20 0.35
CNR1 P21554 1/20 0.35
GLA P06280 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016921 0.92 ADORA2B (0.41) LMNAHTTPARP1NR3C1TPH1
SCHEMBL4295147 0.88 MAOB (0.40) LMNAHTTGAASMN1; SMN2PARP1
SCHEMBL4018480 0.78 TPH1 (0.50) HTTKDM4EALDH1A1HSD17B10SMN1; SMN2
SCHEMBL4016181 0.76 MEN1 (0.42) LMNAHTTALDH1A1HPGD
SCHEMBL5509419 0.74 ADORA3 (0.44) LMNAHTTKDM4EALDH1A1GAA
SCHEMBL4014400 0.73 ADORA2A (0.41) PARP1
SCHEMBL4284406 0.73 NOD1 (0.39) LMNAHTTKDM4EALDH1A1HSD17B10
SCHEMBL5061625 0.73 TPH1 (0.48) HTTKDM4EALDH1A1SMN1; SMN2TPH1
SCHEMBL4016371 0.68 ADORA2B (0.64)
SCHEMBL1720325 0.68 ADORA3 (0.42) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009088518-A1 A2B ADENOSINE RECEPTOR ANTAGONISTS FOR THE TREATMENT OF CANCER CV THERAPEUTICS, INC. (US) 2009-07-16 WO disclosed