SCHEMBL4026426

SCHEMBL4026426

COc1ccc(C(=O)Nc2ccc(CC(=O)NO)cc2)cc1OC

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.61
KMT2A Q03164 6/20 0.61
PKM P14618 3/20 0.60
ALDH1A1 P00352 2/20 0.60
NR1H4 Q96RI1 1/20 0.59
NPC1 O15118 4/20 0.58
POLB P06746 1/20 0.58
RAB9A P51151 4/20 0.58
MAPT P10636 3/20 0.58
LMNA P02545 1/20 0.58
EPHX2 P34913 1/20 0.57
ROCK2 O75116 1/20 0.57
CYP3A4 P08684 1/20 0.57
NQO2 P16083 1/20 0.56
CASP3 P42574 1/20 0.56
SENP7 Q9BQF6 1/20 0.56
USP2 O75604 1/20 0.56
SMN1; SMN2 Q16637 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC8 Q9BY41 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4020377 0.85 MAPT (0.57) MEN1KMT2AALDH1A1NR1H4NPC1
SCHEMBL4020386 0.85 MAPT (0.59) MEN1KMT2AALDH1A1NPC1POLB
SCHEMBL4024552 0.84 NR1H4 (0.53) MEN1KMT2AALDH1A1NR1H4NPC1
SCHEMBL15480650 0.84 MEN1 (0.70) MEN1KMT2APKMALDH1A1NPC1
SCHEMBL29944952 0.83 ROCK2 (0.66) MEN1KMT2AALDH1A1NR1H4NPC1
SCHEMBL4024140 0.83 HDAC1 (0.57) MEN1KMT2AALDH1A1NR1H4NPC1
SCHEMBL14490974 0.83 NPC1 (0.69) MEN1KMT2AALDH1A1NPC1POLB
SCHEMBL4020644 0.82 HDAC1 (0.58) MAPTLMNASMN1; SMN2HDAC1HDAC6
SCHEMBL21156696 0.80 EPHX2 (0.64) KMT2AALDH1A1POLBMAPTLMNA
SCHEMBL4656274 0.80 NPC1 (0.71) MEN1KMT2AALDH1A1NR1H4NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874722-B1 HYDROXAMIC ACID DERIVATIVES AND THE PREPARATION METHOD THEREOF AMOREPACIFIC CORP (KR) 2015-04-08 EP claimed
US-7485750-B2 Hydroxamic acid derivatives and the preparation method thereof AMOREPACIFIC CORPORATION (KR) 2009-02-03 US claimed
US-20080242730-A1 Hydroxamic Acid Derivatives and the Preparation Method Thereof AMOREPACIFIC CORPORATION (KR) 2008-10-02 US claimed
EP-1874722-A1 HYDROXAMIC ACID DERIVATIVES AND THE PREPARATION METHOD THEREOF Amorepacific Corporation (KR) 2008-01-09 EP claimed
WO-2006118380-A1 HYDROXAMIC ACID DERIVATIVES AND THE PREPARATION METHOD THEREOF AMOREPACIFIC CORPORATION (KR) 2006-11-09 WO claimed
EP-1874722-B1 HYDROXAMIC ACID DERIVATIVES AND THE PREPARATION METHOD THEREOF AMOREPACIFIC CORP (KR) 2015-04-08 EP disclosed
US-7485750-B2 Hydroxamic acid derivatives and the preparation method thereof AMOREPACIFIC CORPORATION (KR) 2009-02-03 US disclosed
US-20080242730-A1 Hydroxamic Acid Derivatives and the Preparation Method Thereof AMOREPACIFIC CORPORATION (KR) 2008-10-02 US disclosed
EP-1874722-A1 HYDROXAMIC ACID DERIVATIVES AND THE PREPARATION METHOD THEREOF Amorepacific Corporation (KR) 2008-01-09 EP disclosed
WO-2006118380-A1 HYDROXAMIC ACID DERIVATIVES AND THE PREPARATION METHOD THEREOF AMOREPACIFIC CORPORATION (KR) 2006-11-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080242730-A1 Hydroxamic Acid Derivatives and the Preparation Method Thereof COL14A1, CUTA, COL2A1 MEN1 4712/4885KMT2A 1541/4885PKM 2574/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.