SCHEMBL4031044

SCHEMBL4031044

Cn1c(-c2sccc2NC(=O)Nc2ccccc2-c2ccccc2)nc(OC(=O)O)c(O)c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 2/20 0.41
RET P07949 1/20 0.39
FLT1 P17948 1/20 0.39
KDR P35968 1/20 0.39
MAPK14 Q16539 1/20 0.39
PDE10A Q9Y233 1/20 0.37
CHRM3 P20309 8/20 0.36
TSHR P16473 2/20 0.36
HSD17B10 Q99714 2/20 0.36
USP2 O75604 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
CHRM2 P08172 2/20 0.35
CHRM1 P11229 2/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
ERCC1 P07992 1/20 0.35
FEN1 P39748 1/20 0.35
ERCC4 Q92889 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4031565 0.89 CXCR2 (0.39) MAPK14POLBMAPTALDH1A1LMNA
SCHEMBL4030887 0.86 ERCC1 (0.51) NTRK1RETFLT1KDRMAPK14
SCHEMBL4027166 0.85 MEN1 (0.37) HTTALDH1A1ERCC1FEN1ERCC4
SCHEMBL4028019 0.84 FEN1 (0.39) HSD17B10ERCC1FEN1ERCC4
SCHEMBL4026648 0.83 NTRK1 (0.44) NTRK1RETFLT1KDRMAPK14
SCHEMBL4032051 0.82 RAB9A (0.40) TSHRHSD17B10MAPTALDH1A1
SCHEMBL4028505 0.79 ALDH1A1 (0.38) MAPTHTTALDH1A1ERCC1FEN1
SCHEMBL4026226 0.79 MAOB (0.38) TSHRHSD17B10MAPTHTTALDH1A1
SCHEMBL4027676 0.78 MAPK8 (0.40) HSD17B10MAPTALDH1A1
SCHEMBL4028369 0.78 MEN1 (0.43) MAPTHTTALDH1A1ERCC1FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1470113-B1 PYRIMIDINONE VIRAL POLYMERASE INHIBITORS ANGELETTI P IST RICHERCHE BIO (IT) 2009-01-07 EP claimed