SCHEMBL4031683

SCHEMBL4031683

Cc1noc(-c2ccc(C#N)cc2)c1N(C(=O)O)C(c1ccccc1)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.43
S1PR4 O95977 2/20 0.38
S1PR3 Q99500 2/20 0.38
EP300 Q09472 5/20 0.37
ALDH1A1 P00352 2/20 0.36
LPAR1 Q92633 2/20 0.36
LPAR3 Q9UBY5 1/20 0.36
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
BRD4 O60885 2/20 0.35
PKM P14618 1/20 0.34
MLYCD O95822 1/20 0.34
PTPN5 P54829 1/20 0.34
PRSS1 P07477 1/20 0.34
CTSG P08311 1/20 0.34
CTRB1 P17538 1/20 0.34
CMA1 P23946 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4031919 0.85 TRPA1 (0.50) TRPA1S1PR4S1PR3EP300ALDH1A1
SCHEMBL4030341 0.84 LPAR1 (0.39) S1PR3ALDH1A1LPAR1LPAR3
SCHEMBL4036790 0.77 TRPA1 (0.46) TRPA1EP300ALDH1A1LPAR1LPAR3
SCHEMBL4033561 0.73 LPAR1 (0.42) TRPA1ALDH1A1LPAR1LPAR3
SCHEMBL4028121 0.73 LPAR1 (0.44) TRPA1ALDH1A1LPAR1LPAR3
SCHEMBL4030691 0.73 LPAR1 (0.41) LPAR1LPAR3
SCHEMBL4037774 0.73 LPAR1 (0.33) S1PR3LPAR1MLYCD
SCHEMBL4035140 0.72 KMT2A (0.44)
SCHEMBL4031685 0.72 LPAR1 (0.59) TRPA1S1PR4S1PR3EP300ALDH1A1
SCHEMBL4036870 0.68 MAPK1 (0.42) ALDH1A1LPAR1LPAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed