SCHEMBL4032967

SCHEMBL4032967

Cc1ccc(Sc2c(OC(N)=O)[nH]c3cccnc23)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
GSK3B P49841 1/20 0.38
ADK P55263 1/20 0.38
TGFBR1 P36897 1/20 0.37
PDE9A O76083 1/20 0.37
RAB9A P51151 4/20 0.36
NPC1 O15118 3/20 0.36
SLC6A4 P31645 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
LMNA P02545 2/20 0.35
MAPT P10636 2/20 0.35
HTT P42858 2/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
PDE5A O76074 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4034008 0.90 LMNA (0.37) GSK3BADKTGFBR1LMNAKMT2A
SCHEMBL4035502 0.89 TUBB4A (0.39) SMN1; SMN2ALDH1A1SLC6A4PTGDR2LMNA
SCHEMBL4035489 0.88 SLC6A4 (0.43) SMN1; SMN2ALDH1A1GAATGFBR1RAB9A
SCHEMBL4033192 0.88 PKN1 (0.38) KMT2AMEN1PDE5A
SCHEMBL4043268 0.88 PKN1 (0.36) SMN1; SMN2TGFBR1RAB9ANPC1MAPT
SCHEMBL4039619 0.84 MAPT (0.46) SMN1; SMN2ALDH1A1GAARAB9ANPC1
SCHEMBL4036107 0.83 PDE5A (0.36) ALDH1A1GSK3BADKTGFBR1HTT
SCHEMBL2053135 0.82 SMN1; SMN2 (0.43) SMN1; SMN2ALDH1A1GAATGFBR1PDE9A
SCHEMBL4036370 0.82 PARP1 (0.37) ALDH1A1TGFBR1KMT2AMEN1PDE5A
SCHEMBL4036538 0.81 JAK2 (0.48) ALDH1A1TGFBR1RAB9ANPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747220-B1 SUBSTITUTED 1H-PYRROLO[3,2-B, 3,2-C, AND 2,3-C]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2009-04-15 EP claimed