SCHEMBL4036022

SCHEMBL4036022

NC(=O)Oc1[nH]c2cnccc2c1Sc1ccccc1C(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2 P11137 1/20 0.39
LMNA P02545 2/20 0.38
MAPK1 P28482 1/20 0.38
KIF11 P52732 1/20 0.35
CHUK O15111 3/20 0.35
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
IKBKB O14920 1/20 0.35
AURKA O14965 1/20 0.35
PIM1 P11309 1/20 0.35
TOP1 P11387 1/20 0.35
GABRA1 P14867 1/20 0.35
IDO1 P14902 1/20 0.35
HPGD P15428 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
MAOA P21397 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043021 0.88 MAP2 (0.38) MAP2MAPK1KIF11CHUKKDM4E
SCHEMBL2052333 0.84 MAP2 (0.52) MAP2LMNAMAPK1KIF11CHUK
SCHEMBL4038766 0.83 TUBB4A (0.45) MAP2CHUKKDM4EALDH1A1SMN1; SMN2
SCHEMBL4038757 0.82 MAP2 (0.46) MAP2LMNACHUKKDM4EALDH1A1
SCHEMBL4039379 0.80 CHUK (0.42) MAP2CHUKKDM4EALDH1A1SMN1; SMN2
SCHEMBL4038003 0.80 PARP1 (0.39) LMNAKIF11KDM4EPARP1RBP4
SCHEMBL3270325 0.77 KDM4E (0.35) LMNAKDM4EALDH1A1HPGDPARP1
SCHEMBL4043016 0.77 ROCK2 (0.40) MAP2CHUKSMN1; SMN2PIM1KDM5A
SCHEMBL4035359 0.74 CSNK2A2 (0.42) MAP2LMNACHUKALDH1A1ICOSLG
SCHEMBL4042867 0.73 TUBB4A (0.46) CHUKICOSLGICOSROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1747220-B1 SUBSTITUTED 1H-PYRROLO[3,2-B, 3,2-C, AND 2,3-C]PYRIDINE-2-CARBOXAMIDES AND RELATED ANALOGS AS INHIBITORS OF CASEIN KINASE I EPSILON AVENTIS PHARMA INC (US) 2009-04-15 EP claimed