SCHEMBL4037073

SCHEMBL4037073

CC(C)Oc1ccc(C#CCCCC#N)cc1C(=O)N[C@](C)(O)Cc1c[nH]c2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.39
MEN1 O00255 3/20 0.39
CYP2D6 P10635 6/20 0.39
CTSL P07711 2/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
CDK2 P24941 1/20 0.38
TACR1 P25103 4/20 0.38
SLC22A1 O15245 1/20 0.38
CTSC P53634 1/20 0.36
TACR3 P29371 1/20 0.35
ALOX5 P09917 1/20 0.35
EPHX2 P34913 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4035462 0.91 KMT2A (0.41) KMT2AMEN1CYP2D6CDK2TACR1
SCHEMBL4033975 0.90 MAPT (0.39) KMT2AMEN1CYP2D6TACR1MAPT
SCHEMBL4038448 0.87 KMT2A (0.42) KMT2AMEN1CYP2D6CDK2TACR1
SCHEMBL3943652 0.84 CTSL (0.41) KMT2AMEN1CTSLCTSSCTSK
SCHEMBL4031864 0.82 MAPT (0.40) KMT2AMEN1TACR1MAPT
SCHEMBL4034270 0.82 KMT2A (0.46) KMT2AMEN1TACR1TACR3MAPT
SCHEMBL4037068 0.80 KMT2A (0.40) KMT2AMEN1CTSLCTSSCTSK
SCHEMBL4037079 0.80 KMT2A (0.40) KMT2AMEN1CTSLCTSSCTSK
SCHEMBL13904509 0.79 MMP9 (0.43) KMT2AMEN1CYP2D6TACR1TACR3
SCHEMBL3947792 0.79 MMP9 (0.43) KMT2AMEN1CYP2D6TACR1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2019102-A1 Alkylacetylene substituted Acyltryptophanols Bayer Schering Pharma AG (DE) 2009-01-28 EP disclosed