SCHEMBL4033975

SCHEMBL4033975

CNC(=O)CCCC#Cc1ccc(OC(C)C)c(C(=O)N[C@](C)(O)Cc2c[nH]c3ccccc23)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.39
KMT2A Q03164 7/20 0.38
MEN1 O00255 6/20 0.38
HCRTR1 O43613 1/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NMBR P28336 1/20 0.37
HPGD P15428 2/20 0.37
TACR1 P25103 1/20 0.36
CYP2D6 P10635 4/20 0.36
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
RECQL P46063 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35
TDP1 Q9NUW8 2/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4037073 0.90 KMT2A (0.39) MAPTKMT2AMEN1TACR1CYP2D6
SCHEMBL4035462 0.89 KMT2A (0.41) MAPTKMT2AMEN1KDM4EL3MBTL1
SCHEMBL4038448 0.85 KMT2A (0.42) MAPTKMT2AMEN1KDM4EALDH1A1
SCHEMBL3939353 0.84 MEN1 (0.42) MAPTKMT2AMEN1HCRTR1KDM4E
SCHEMBL4033976 0.81 MEN1 (0.39) MAPTKMT2AMEN1HCRTR1KDM4E
SCHEMBL4033972 0.81 MEN1 (0.39) MAPTKMT2AMEN1HCRTR1KDM4E
SCHEMBL4031864 0.81 MAPT (0.40) MAPTKMT2AMEN1NMBRTACR1
SCHEMBL4033963 0.80 MPO (0.46) CYP2D6
SCHEMBL4034270 0.80 KMT2A (0.46) MAPTKMT2AMEN1KDM4EALDH1A1
SCHEMBL3945226 0.80 MMP9 (0.40) MAPTKMT2AMEN1HCRTR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2019102-A1 Alkylacetylene substituted Acyltryptophanols Bayer Schering Pharma AG (DE) 2009-01-28 EP disclosed