SCHEMBL4038893

SCHEMBL4038893

NC(=O)c1ccccc1CCCCNC[C@@H](O)[CH]Cc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A5 Q9Y345 6/20 0.39
ABCB1 P08183 5/20 0.37
CYP2D6 P10635 4/20 0.37
LMNA P02545 4/20 0.37
ADRB2 P07550 4/20 0.37
ADRB1 P08588 4/20 0.37
CYP1A2 P05177 3/20 0.37
ADRA1A P35348 3/20 0.37
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
HTR2B P41595 2/20 0.37
SLC6A3 Q01959 2/20 0.37
SIGMAR1 Q99720 2/20 0.37
THPO P40225 2/20 0.37
HIF1A Q16665 2/20 0.37
ADRA2A P08913 2/20 0.37
ADRA1D P25100 2/20 0.37
ADRA1B P35368 2/20 0.37
ADRB3 P13945 2/20 0.37
ADRA2C P18825 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049170 0.97 MPO (0.39) SLC6A5ABCB1CYP2D6LMNAADRB2
SCHEMBL4044662 0.92 ABCB1 (0.39) ABCB1CYP2D6LMNAADRB2ADRB1
SCHEMBL4036513 0.78 RPS6KB1 (0.40) ABCB1CYP2D6LMNAADRB2ADRB1
SCHEMBL4039140 0.77 ABCB1 (0.47) ABCB1CYP2D6LMNAADRB2ADRB1
SCHEMBL4047555 0.77 SIRT1 (0.38) SLC6A5CYP2D6LMNAADRB2ADRB1
SCHEMBL4045617 0.76 ADRB1 (0.36) ABCB1CYP2D6LMNAADRB2ADRB1
SCHEMBL11322428 0.75 KDM4E (0.43) CYP2D6LMNAADRB2ADRB1CYP1A2
SCHEMBL4044458 0.75 ADRB2 (0.39) ABCB1CYP2D6LMNAADRB2ADRB1
Methylamine SCHEMBL28758829 0.74 SIGMAR1 (0.48) SIGMAR1SMN1; SMN2ALDH1A1HPGDMEN1
SCHEMBL29410986 0.74 BID (0.51) SLC6A5LMNAADRB2ADRA1ASLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed