SCHEMBL4044458

SCHEMBL4044458

NC(=O)Oc1ccccc1CCNC[C@H](O)[CH]Cc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.39
ADRB1 P08588 6/20 0.39
ADRB3 P13945 6/20 0.39
ABCB1 P08183 5/20 0.39
LMNA P02545 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP3A4 P08684 2/20 0.39
KCNK3 O14649 1/20 0.39
SLC22A1 O15245 1/20 0.39
ABCC9 O60706 1/20 0.39
KCNK2 O95069 1/20 0.39
ABCB11 O95342 1/20 0.39
ADRA2C P18825 1/20 0.39
SLC6A2 P23975 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
SLC6A4 P31645 1/20 0.39
ADRA1A P35348 1/20 0.39
HTR2B P41595 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4037688 0.83 KDM4E (0.46) ADRB2ADRB1ADRB3SMN1; SMN2KMT2A
SCHEMBL4044662 0.82 ABCB1 (0.39) ADRB2ADRB1ADRB3ABCB1LMNA
SCHEMBL4042381 0.81 ADRB2 (0.59) ADRB2ADRB1ADRB3LMNACYP2D6
SCHEMBL4041765 0.81 ADRB3 (0.46) ADRB2ADRB1ADRB3CYP2D6KMT2A
SCHEMBL4045617 0.78 ADRB1 (0.36) ADRB2ADRB1ADRB3ABCB1LMNA
SCHEMBL4049170 0.76 MPO (0.39) ADRB2ADRB1ADRB3ABCB1LMNA
SCHEMBL4038893 0.75 SLC6A5 (0.39) ADRB2ADRB1ADRB3ABCB1LMNA
SCHEMBL4048154 0.74 BCHE (0.43) KMT2AMEN1
SCHEMBL4041577 0.72 ALDH1A1 (0.38) ADRA2CKMT2AMEN1METAP2METAP1
SCHEMBL4036513 0.71 RPS6KB1 (0.40) ADRB2ADRB1ADRB3ABCB1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2051967-A1 BENZIMIDAZOLE DERIVATIVES USEFUL IN TREATMENT OF VALLINOID RECEPTOR TRPV1 RELATED DISORDERS AstraZeneca AB (SE) 2009-04-29 EP claimed
WO-2008018827-A1 BENZIMIDAZOLE DERIVATIVES USEFUL IN TREATMENT OF VALLINOID RECEPTOR TRPV1 RELATED DISORDERS ASTRAZENECA AB (SE) 2008-02-14 WO claimed