SCHEMBL4039771

SCHEMBL4039771

CCCC(NC(=O)Oc1ccc2ncccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1ccccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.38
PREP P48147 2/20 0.35
FAP Q12884 2/20 0.35
CTSK P43235 4/20 0.33
NR2F2 P24468 2/20 0.33
RAB9A P51151 2/20 0.33
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33
ELANE P08246 1/20 0.32
ALOX5 P09917 1/20 0.32
ITGB2 P05107 2/20 0.32
ICAM1 P05362 2/20 0.32
ITGAL P20701 2/20 0.32
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32
CTSS P25774 1/20 0.32
GALR3 O60755 1/20 0.31
ATM Q13315 1/20 0.31
MAPT P10636 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045026 0.95 CTSK (0.36) ALDH1A1PREPFAPCTSKELANE
SCHEMBL4041598 0.93 CTSK (0.40) ALDH1A1CTSKELANECTSLCTSB
SCHEMBL4046799 0.90 ALDH1A1 (0.39) ALDH1A1PREPFAPCTSKCTSL
SCHEMBL4047431 0.90 ALDH1A1 (0.37) ALDH1A1PREPFAPNR2F2RAB9A
SCHEMBL4043139 0.89 ELANE (0.37) ALDH1A1PREPFAPCTSKELANE
SCHEMBL4043678 0.88 ALDH1A1 (0.38) ALDH1A1PREPFAPCTSKNR2F2
SCHEMBL4048179 0.88 TSHR (0.36) ALDH1A1PREPFAPRAB9AELANE
SCHEMBL4051956 0.87 CTSK (0.41) CTSKELANECTSLCTSBCTSS
SCHEMBL4044622 0.87 CTSK (0.38) PREPFAPCTSKELANECTSL
SCHEMBL4045022 0.87 CTSK (0.35) PREPFAPCTSKELANECTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506175-B1 N-SUBSTITUTED TRICYCLIC 3-AMINOPYRAZOLES AS PDGF RECEPTOR INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2009-04-01 EP disclosed