SCHEMBL4047431

SCHEMBL4047431

CCCC(NC(=O)Oc1ccc2ncccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
SMYD3 Q9H7B4 2/20 0.34
GPR132 Q9UNW8 3/20 0.33
NAMPT P43490 1/20 0.33
TNF P01375 1/20 0.33
MAPK1 P28482 1/20 0.33
NOD2 Q9HC29 1/20 0.33
NOD1 Q9Y239 1/20 0.33
PREP P48147 1/20 0.33
FAP Q12884 1/20 0.33
NR2F2 P24468 2/20 0.32
RAB9A P51151 1/20 0.32
GPBAR1 Q8TDU6 1/20 0.32
KMT2A Q03164 1/20 0.32
PPARG P37231 1/20 0.32
PPARA Q07869 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047844 0.94 SMYD3 (0.35) SMYD3
SCHEMBL4041373 0.93 CTSK (0.38) ALDH1A1SMYD3NAMPTTNFMAPK1
SCHEMBL4046989 0.90 ALDH1A1 (0.38) ALDH1A1MAPK1PREPFAPNR2F2
SCHEMBL4039771 0.90 ALDH1A1 (0.38) ALDH1A1PREPFAPNR2F2RAB9A
SCHEMBL4044339 0.89 ALDH1A1 (0.37) ALDH1A1GPR132PREPFAPNR2F2
SCHEMBL4043998 0.88 FKBP1A (0.37) SMYD3NAMPT
SCHEMBL4044443 0.88 ALDH1A1 (0.38) ALDH1A1GPR132TNFMAPK1NOD2
SCHEMBL4043650 0.87 BMP1 (0.36) ALDH1A1SMYD3NAMPTKMT2A
SCHEMBL4050147 0.86 CTSK (0.40) SMYD3
SCHEMBL4046799 0.86 ALDH1A1 (0.39) ALDH1A1PREPFAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed