SCHEMBL4043678

SCHEMBL4043678

CCCC(NC(=O)Oc1ccc2ncccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1ccccn1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
PREP P48147 1/20 0.35
FAP Q12884 1/20 0.35
RAB9A P51151 4/20 0.34
NR2F2 P24468 2/20 0.34
PPARG P37231 1/20 0.34
PPARA Q07869 1/20 0.34
MC4R P32245 1/20 0.34
MC3R P41968 1/20 0.34
MC1R Q01726 1/20 0.34
LMNA P02545 2/20 0.33
ALOX5 P09917 1/20 0.33
CTSK P43235 3/20 0.33
GALR3 O60755 1/20 0.32
ATM Q13315 1/20 0.32
MAPT P10636 3/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 2/20 0.32
HDAC1 Q13547 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047535 0.95 MC4R (0.38) PREPFAPMC4RMC3RMC1R
SCHEMBL4043226 0.93 CTSK (0.40) ALDH1A1RAB9ALMNACTSKCTSL
SCHEMBL4046799 0.90 ALDH1A1 (0.39) ALDH1A1PREPFAPCTSKCTSL
SCHEMBL4044339 0.90 ALDH1A1 (0.37) ALDH1A1PREPFAPRAB9ANR2F2
SCHEMBL4052303 0.89 CTSK (0.35) PREPFAPMC4RMC3RMC1R
SCHEMBL4049188 0.89 CTSK (0.40) ALDH1A1PREPFAPRAB9ANR2F2
SCHEMBL4039771 0.88 ALDH1A1 (0.38) ALDH1A1PREPFAPRAB9ANR2F2
SCHEMBL4046061 0.88 LMNA (0.36) ALDH1A1PREPFAPRAB9ALMNA
SCHEMBL4043256 0.87 CTSK (0.41) ALDH1A1MC4RMC3RMC1RCTSK
SCHEMBL4043203 0.87 CTSK (0.35) ALDH1A1PREPFAPRAB9AMC4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed