SCHEMBL4040431

SCHEMBL4040431

CCCC(NC(=O)Oc1oc2ccccc2c1C)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.37
CHRNA7 P36544 1/20 0.37
CHRNA4 P43681 1/20 0.37
GAA P10253 2/20 0.36
PREP P48147 2/20 0.35
FAP Q12884 2/20 0.35
CTSK P43235 4/20 0.34
NPSR1 Q6W5P4 3/20 0.33
USP2 O75604 3/20 0.33
LMNA P02545 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
TSHR P16473 1/20 0.33
PAX8 Q06710 1/20 0.32
IGLV6-57 P01721 1/20 0.32
ACACB O00763 1/20 0.32
PSMB8 P28062 1/20 0.32
PSMB5 P28074 1/20 0.32
HTT P42858 2/20 0.31
P2RX7 Q99572 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050081 0.93 CTSK (0.42) CHRNB2CHRNA7CHRNA4GAACTSK
SCHEMBL4041842 0.92 CHRNB2 (0.37) CHRNB2CHRNA7CHRNA4GAACTSK
SCHEMBL4044961 0.89 CHRNB2 (0.35) CHRNB2CHRNA7CHRNA4GAACTSK
SCHEMBL4048128 0.88 CHRNB2 (0.36) CHRNB2CHRNA7CHRNA4GAAPREP
SCHEMBL4046786 0.86 CHRNB2 (0.36) CHRNB2CHRNA7CHRNA4PREPFAP
SCHEMBL4042714 0.85 SMN1; SMN2 (0.36) CHRNB2CHRNA7CHRNA4GAAPREP
SCHEMBL4047771 0.84 CTSK (0.39) CHRNA7CTSKACACB
SCHEMBL4046502 0.84 PREP (0.34) CHRNB2CHRNA7CHRNA4GAAPREP
SCHEMBL4050441 0.84 CTSK (0.39) PREPFAPCTSKSMN1; SMN2HTT
SCHEMBL4041663 0.84 CTSK (0.35) PREPFAPCTSKUSP2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed