SCHEMBL4046786

SCHEMBL4046786

CCCC(NC(=O)Oc1cc2ccccc2o1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.36
CHRNA7 P36544 4/20 0.36
CHRNA4 P43681 4/20 0.36
KCNH2 Q12809 1/20 0.36
CTSK P43235 3/20 0.35
PSMB5 P28074 1/20 0.34
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 1/20 0.34
PAX8 Q06710 1/20 0.33
GFER P55789 1/20 0.33
NAMPT P43490 1/20 0.33
PREP P48147 1/20 0.33
FAP Q12884 1/20 0.33
MKNK1 Q9BUB5 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HTRA1 Q92743 1/20 0.33
POLB P06746 1/20 0.32
HTT P42858 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042383 0.93 CTSK (0.42) CHRNB2CHRNA7CHRNA4KCNH2CTSK
SCHEMBL4044034 0.92 CHRNB2 (0.41) CHRNB2CHRNA7CHRNA4ALDH1A1KDM4E
SCHEMBL4046927 0.89 CHRNA7 (0.41) CHRNB2CHRNA7CHRNA4CTSKALDH1A1
SCHEMBL4043031 0.88 HTRA1 (0.37) CHRNA7CTSKPAX8NAMPTHTRA1
SCHEMBL4046863 0.88 SMYD3 (0.35) CHRNB2CHRNA7CHRNA4KCNH2CTSK
SCHEMBL4041663 0.87 CTSK (0.35) CTSKPAX8PREPFAPSMN1; SMN2
SCHEMBL4043616 0.86 CTSK (0.35) CTSKALDH1A1PAX8PREPFAP
SCHEMBL4040431 0.86 CHRNB2 (0.37) CHRNB2CHRNA7CHRNA4CTSKPSMB5
SCHEMBL4041999 0.85 HSD17B10 (0.36) CTSKALDH1A1KDM4EPREPFAP
SCHEMBL4041238 0.85 CHRNB2 (0.36) CHRNB2CHRNA7CHRNA4CTSKPAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed