SCHEMBL4041842

SCHEMBL4041842

Cc1c(OC(=O)NC(CC2CC2)C(=O)N2CCC3C2C(=O)CN3C(=O)Cc2cccnc2)oc2ccccc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.37
CHRNA7 P36544 2/20 0.37
CHRNA4 P43681 2/20 0.37
GAA P10253 2/20 0.36
CTSK P43235 2/20 0.34
CTSV O60911 2/20 0.33
CTSL P07711 2/20 0.33
CTSS P25774 2/20 0.33
HTRA1 Q92743 1/20 0.33
USP2 O75604 3/20 0.32
LMNA P02545 3/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
NPSR1 Q6W5P4 2/20 0.32
TSHR P16473 1/20 0.32
PAX8 Q06710 1/20 0.32
PSMB8 P28062 1/20 0.32
PSMB5 P28074 1/20 0.32
HTT P42858 2/20 0.31
TP53 P04637 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050081 0.93 CTSK (0.42) CHRNB2CHRNA7CHRNA4GAACTSK
SCHEMBL4040431 0.92 CHRNB2 (0.37) CHRNB2CHRNA7CHRNA4GAACTSK
SCHEMBL4044961 0.89 CHRNB2 (0.35) CHRNB2CHRNA7CHRNA4GAACTSK
SCHEMBL4049249 0.88 CHRNB2 (0.36) CHRNB2CHRNA7CHRNA4GAACTSV
SCHEMBL4042994 0.84 CTSS (0.35) CHRNB2CHRNA7CHRNA4GAACTSK
SCHEMBL4042558 0.84 CTSK (0.39) CTSKCTSVCTSLCTSSSMN1; SMN2
SCHEMBL4041874 0.82 CHRNB2 (0.37) CHRNB2CHRNA7CHRNA4GAAUSP2
SCHEMBL6233220 0.81 CHRNB2 (0.48) CHRNB2CHRNA7CHRNA4GAACTSK
SCHEMBL4043880 0.81 CHRNB2 (0.41) CHRNB2CHRNA7CHRNA4GAACTSK
SCHEMBL4044165 0.81 CTSK (0.38) CHRNB2CHRNA7CHRNA4GAACTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed