SCHEMBL4040539

SCHEMBL4040539

O=C(NC(Cc1ccc(F)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1ccccn1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MC4R P32245 2/20 0.41
MC3R P41968 2/20 0.41
MC1R Q01726 2/20 0.41
P2RX7 Q99572 2/20 0.35
GPR34 Q9UPC5 1/20 0.35
PSMB5 P28074 2/20 0.34
ITGA4 P13612 5/20 0.34
ITGB7 P26010 5/20 0.34
SCN9A Q15858 3/20 0.34
ITGB1 P05556 2/20 0.34
CTSK P43235 2/20 0.34
HTRA1 Q92743 1/20 0.33
USP30 Q70CQ3 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044814 0.94 FNTA (0.35) MC4RMC3RMC1RPSMB5ITGA4
SCHEMBL4045924 0.93 USP30 (0.40) MC4RMC3RMC1RITGA4ITGB7
SCHEMBL6210192 0.90 CTSK (0.43) MC4RMC3RMC1RPSMB5ITGB1
SCHEMBL4043350 0.89 HTRA1 (0.35) MC4RMC3RMC1RPSMB5ITGA4
SCHEMBL4052754 0.88 CTSK (0.42) MC4RMC3RMC1RP2RX7GPR34
SCHEMBL4045521 0.88 CTSK (0.43) SCN9ACTSK
SCHEMBL4043465 0.88 MC4R (0.41) MC4RMC3RMC1RP2RX7ITGA4
SCHEMBL4049324 0.88 MC4R (0.37) MC4RMC3RMC1RP2RX7GPR34
SCHEMBL4052303 0.88 CTSK (0.35) MC4RMC3RMC1RCTSK
SCHEMBL6210306 0.86 CTSK (0.43) MC4RMC3RMC1RITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed