SCHEMBL4049324

SCHEMBL4049324

O=C(NC(Cc1ccc(F)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1ccccn1)Oc1ccc(-c2ccccc2)cc1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MC4R P32245 3/20 0.37
MC3R P41968 3/20 0.37
MC1R Q01726 3/20 0.37
ITGA4 P13612 2/20 0.37
ITGB7 P26010 2/20 0.37
ELANE P08246 1/20 0.35
P2RX7 Q99572 2/20 0.35
GPR34 Q9UPC5 1/20 0.35
PAX8 Q06710 1/20 0.34
CTSK P43235 2/20 0.34
SCN9A Q15858 2/20 0.33
ITGB1 P05556 2/20 0.33
ITGB3 P05106 1/20 0.33
ITGAV P06756 1/20 0.33
ITGA5 P08648 1/20 0.33
XIAP P98170 1/20 0.33
FPR1 P21462 2/20 0.32
FPR2 P25090 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044539 0.94 ITGA4 (0.36) ITGA4ITGB7ELANEP2RX7CTSK
SCHEMBL4051785 0.93 ITGA4 (0.39) ITGA4ITGB7ELANECTSKITGB3
SCHEMBL6211121 0.90 CTSK (0.43) MC4RMC3RMC1RITGA4ITGB7
SCHEMBL4046932 0.89 GPR132 (0.35) ITGA4ITGB7ELANECTSKITGB3
SCHEMBL4050328 0.89 SCN9A (0.39) MC4RMC3RMC1RITGA4ITGB7
SCHEMBL4045311 0.88 CTSK (0.43) ELANECTSK
SCHEMBL4040539 0.88 MC4R (0.41) MC4RMC3RMC1RITGA4ITGB7
SCHEMBL4043139 0.88 ELANE (0.37) ITGA4ITGB7ELANECTSK
SCHEMBL4041436 0.84 ALDH1A1 (0.39) MC4RMC3RMC1RITGA4ITGB7
SCHEMBL4052754 0.84 CTSK (0.42) MC4RMC3RMC1RP2RX7GPR34

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed