SCHEMBL4041104

SCHEMBL4041104

CC(C)(C)OC(=O)On1nc(N)c2cc(NC(=O)Cc3cccc(O)c3)ccc21

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ANO1 Q5XXA6 2/20 0.44
NLRP3 Q96P20 13/20 0.42
RIPK1 Q13546 2/20 0.37
NPY5R Q15761 1/20 0.37
RORC P51449 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL922192 0.85 ANO1 (0.46) ANO1NLRP3RIPK1NPY5R
SCHEMBL5568675 0.78 NLRP3 (0.44) ANO1NLRP3NPY5R
SCHEMBL3933572 0.78 ROCK2 (0.49)
SCHEMBL4035945 0.74 NR1H2 (0.38) RIPK1
SCHEMBL3933114 0.74 NR1H2 (0.36)
SCHEMBL3935784 0.72 KMT2A (0.40) ANO1
SCHEMBL4035815 0.69 JAK2 (0.55) NLRP3
Hydrochloric Acid SCHEMBL921534 0.69 JAK2 (0.54) NLRP3
SCHEMBL1228644 0.68 ROCK2 (0.53)
SCHEMBL5102413 0.65 GAA (0.66) NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765788-B1 3-AMINOINDAZOLE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF SGK-ASSOCIATED DISEASES MERCK PATENT GMBH (DE) 2009-06-03 EP disclosed
EP-1765788-A2 3-AMINOINDAZOLE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF SGK-ASSOCIATED DISEASES MERCK PATENT GmbH (DE) 2007-03-28 EP disclosed
WO-2005123688-A2 3-AMINOINDAZOLES MERCK PATENT GMBH (DE) 2005-12-29 WO disclosed