SCHEMBL4041825

SCHEMBL4041825

O=C(O)CN1C(=O)C(Cc2ccccc2)NC12CCN(C(=S)NCC1CCCCC1)CC2

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.43
ALDH1A1 P00352 4/20 0.42
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CCR5 P51681 2/20 0.39
KMT2A Q03164 3/20 0.38
MEN1 O00255 1/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
ACE P12821 4/20 0.37
KDM4E B2RXH2 1/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3920433 0.86 ATM (0.40) NPSR1ALDH1A1CCR5KMT2AMEN1
SCHEMBL3917759 0.83 NPSR1 (0.39) NPSR1ALDH1A1LMNASMN1; SMN2CCR5
SCHEMBL2943556 0.82 LMNA (0.49) ALDH1A1LMNASMN1; SMN2CCR5KMT2A
SCHEMBL4041819 0.81 CCR5 (0.37) ALDH1A1LMNASMN1; SMN2CCR5KMT2A
SCHEMBL2941205 0.80 MEN1 (0.44) ALDH1A1LMNASMN1; SMN2KMT2AMEN1
SCHEMBL2932813 0.79 MEN1 (0.43) ALDH1A1LMNASMN1; SMN2KMT2AMEN1
SCHEMBL4038265 0.79 KDM4E (0.37) LMNACCR5KMT2AMEN1GAA
SCHEMBL2938912 0.76 CYP3A4 (0.42) ALDH1A1LMNASMN1; SMN2CCR5KMT2A
SCHEMBL2941530 0.75 HPGD (0.43) NPSR1ALDH1A1LMNASMN1; SMN2KMT2A
SCHEMBL2934783 0.74 CCR5 (0.40) ALDH1A1LMNASMN1; SMN2CCR5KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed