SCHEMBL4038265

SCHEMBL4038265

CCOC(=O)NC(=S)N1CCC2(CC1)NC(Cc1ccccc1)C(=O)N2CC(=O)O

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.37
GAA P10253 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.36
CCR5 P51681 2/20 0.36
ABCB11 O95342 1/20 0.35
ACE P12821 1/20 0.35
AGTR2 P50052 1/20 0.35
PDE3A Q14432 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CYP3A4 P08684 1/20 0.35
LMNA P02545 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CXCR3 P49682 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3925416 0.85 KDM4E (0.36) KDM4EL3MBTL1TDP1LMNAMEN1
SCHEMBL3928453 0.84 KDM4E (0.36) KDM4EGAAL3MBTL1TDP1LMNA
SCHEMBL4037263 0.83 ALDH1A1 (0.32)
SCHEMBL4041825 0.79 NPSR1 (0.43) KDM4EGAACCR5ACETDP1
SCHEMBL3917023 0.79 KDM4E (0.48) KDM4EGAATDP1LMNAMEN1
SCHEMBL2934783 0.78 CCR5 (0.40) GAACCR5LMNAMEN1KMT2A
SCHEMBL4032393 0.78 SIGMAR1 (0.39) KDM4EMEN1KMT2ACXCR3
SCHEMBL2938912 0.78 CYP3A4 (0.42) KDM4EGAACCR5CYP3A4LMNA
SCHEMBL2932813 0.77 MEN1 (0.43) KDM4EL3MBTL1LMNAMEN1KMT2A
SCHEMBL2940845 0.76 GRM5 (0.47) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed