SCHEMBL4041819

SCHEMBL4041819

CN(C(=S)N1CCC2(CC1)NC(Cc1ccccc1)C(=O)N2CC(=O)O)C1CCCCC1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 5/20 0.37
ALDH1A1 P00352 3/20 0.37
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ACE P12821 3/20 0.34
ABCC1 P33527 1/20 0.34
GAA P10253 1/20 0.34
RECQL P46063 1/20 0.34
USP19 O94966 2/20 0.34
ATM Q13315 1/20 0.33
USP2 O75604 1/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3917757 0.84 CCR5 (0.35) CCR5ALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL2941205 0.81 MEN1 (0.44) ALDH1A1LMNASMN1; SMN2MEN1KMT2A
SCHEMBL4041825 0.81 NPSR1 (0.43) CCR5ALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL2932813 0.79 MEN1 (0.43) ALDH1A1LMNASMN1; SMN2MEN1KMT2A
SCHEMBL2943556 0.78 LMNA (0.49) CCR5ALDH1A1LMNASMN1; SMN2KMT2A
SCHEMBL2938912 0.78 CYP3A4 (0.42) CCR5ALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL2934783 0.76 CCR5 (0.40) CCR5ALDH1A1LMNASMN1; SMN2MEN1
SCHEMBL4038265 0.75 KDM4E (0.37) CCR5LMNAMEN1KMT2AACE
SCHEMBL2941530 0.75 HPGD (0.43) ALDH1A1LMNASMN1; SMN2MEN1KMT2A
SCHEMBL2940845 0.74 GRM5 (0.47) ALDH1A1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730144-B1 SUBSTITUTED 1,4,8-TRIAZASPIRO¬4.5 DECAN-2-ONE COMPOUNDS GRUENENTHAL GMBH (DE) 2009-06-10 EP claimed