SCHEMBL4043147

SCHEMBL4043147

CC(C)CC(NC(=O)Oc1ccsc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1ccccn1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.40
KMT2A Q03164 1/20 0.37
ELANE P08246 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.35
MAPK1 P28482 1/20 0.35
CTSL P07711 8/20 0.34
CTSS P25774 7/20 0.34
CTSB P07858 3/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045469 0.92 ELANE (0.37) CTSKKMT2AELANESMN1; SMN2CTSL
SCHEMBL4047831 0.92 PREP (0.35) CTSKKMT2AELANEALDH1A1
SCHEMBL4045653 0.90 CTSS (0.38) CTSKKMT2AELANESMN1; SMN2MAPK1
SCHEMBL4045311 0.89 CTSK (0.43) CTSKKMT2AELANESMN1; SMN2MAPK1
SCHEMBL4046866 0.89 CTSK (0.43) CTSKCTSLCTSSCTSB
SCHEMBL4046882 0.89 CTSK (0.41) CTSKKMT2AELANESMN1; SMN2MAPK1
SCHEMBL4050151 0.88 CTSK (0.41) CTSKKMT2ACTSLCTSSCTSB
SCHEMBL4051956 0.88 CTSK (0.41) CTSKKMT2AELANECTSLCTSS
SCHEMBL4045340 0.88 CTSK (0.40) CTSKKMT2AELANESMN1; SMN2MAPK1
SCHEMBL4042764 0.87 CTSK (0.38) CTSKCTSLCTSSCTSBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed