SCHEMBL4043203

SCHEMBL4043203

CCCC(NC(=O)Oc1cc2ccccc2s1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)C(=O)c1ccccn1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 12/20 0.35
PREP P48147 2/20 0.34
FAP Q12884 2/20 0.34
MC4R P32245 1/20 0.33
MC3R P41968 1/20 0.33
MC1R Q01726 1/20 0.33
CTSL P07711 5/20 0.31
CTSS P25774 5/20 0.31
CTSB P07858 2/20 0.31
CTSV O60911 1/20 0.31
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
CRHBP P24387 1/20 0.30
HTT P42858 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30
CRHR2 Q13324 1/20 0.30
P2RY12 Q9H244 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4048011 0.93 CTSK (0.40) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4044612 0.91 PREP (0.33) CTSKPREPFAPMC4RMC3R
SCHEMBL4043984 0.90 CTSK (0.39) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4047535 0.89 MC4R (0.38) CTSKPREPFAPMC4RMC3R
SCHEMBL4045685 0.88 PREP (0.34) CTSKPREPFAPMC4RMC3R
SCHEMBL4043756 0.88 CTSK (0.40) CTSKPREPFAPMC4RMC3R
SCHEMBL4042570 0.88 CTSK (0.34) CTSKPREPFAPMC4RMC3R
SCHEMBL4045022 0.88 CTSK (0.35) CTSKPREPFAPCTSLCTSS
SCHEMBL4039641 0.88 CTSK (0.34) CTSKPREPFAPP2RY12
SCHEMBL4047432 0.88 ALDH1A1 (0.35) CTSKPREPFAPCTSSALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed