SCHEMBL4043459

SCHEMBL4043459

CC(C[CH]C(=O)N1CCC2C1C(=O)CN2C(=O)c1cc[n+]([O-])cc1)C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.41
ATM Q13315 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31
STAT3 P40763 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049285 0.90 CTSK (0.41) CTSKKDM4E
SCHEMBL4048376 0.88 CTSK (0.51) CTSKALDH1A1
SCHEMBL4044693 0.87 CTSK (0.42) CTSKALDH1A1GAA
SCHEMBL4044452 0.85 CTSK (0.39) CTSK
SCHEMBL4044364 0.84 AKR1C3 (0.31)
SCHEMBL4044247 0.83 CTSK (0.39) CTSKALDH1A1
SCHEMBL4050761 0.81 PIK3CD (0.42) CTSKALDH1A1GAA
SCHEMBL4042992 0.80 CTSK (0.39) CTSKALDH1A1GAA
SCHEMBL4037609 0.80 CTSK (0.31) CTSK
SCHEMBL4042279 0.80 CTSK (0.37) CTSKALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed