SCHEMBL4044596

SCHEMBL4044596

Cc1c(OC(=O)NC2(C(=O)N3CCC4C3C(=O)CN4C(=O)c3ccccn3)CCCCC2)oc2ccccc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.38
CTSS P25774 2/20 0.38
CTSK P43235 2/20 0.38
ALDH1A1 P00352 2/20 0.33
HTT P42858 2/20 0.33
HSD17B10 Q99714 1/20 0.33
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
FAAH O00519 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
RECQL P46063 1/20 0.31
EPHX2 P34913 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
NPC1 O15118 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4044049 0.89 CTSL (0.33) CTSLCTSSCTSKLMNAGAA
SCHEMBL6238275 0.88 CTSL (0.40) CTSLCTSSCTSKALDH1A1HTT
SCHEMBL4041595 0.86 CTSK (0.42) CTSLCTSSCTSK
SCHEMBL4042694 0.84 CTSL (0.34) CTSLCTSSCTSKALDH1A1HSD17B10
SCHEMBL4041874 0.83 CHRNB2 (0.37) HTTLMNAGAATSHRMEN1
SCHEMBL4045681 0.81 LMNA (0.36) CTSLCTSSCTSKALDH1A1HTT
SCHEMBL4047235 0.80 CTSL (0.36) CTSLCTSSCTSKALDH1A1HSD17B10
SCHEMBL4041529 0.80 CTSK (0.47) CTSLCTSSCTSKALDH1A1HSD17B10
SCHEMBL4042558 0.80 CTSK (0.39) CTSLCTSSCTSKALDH1A1HTT
SCHEMBL4050441 0.80 CTSK (0.39) CTSLCTSSCTSKALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed