SCHEMBL4045035

SCHEMBL4045035

CC(C)CC(NC(=O)Oc1ccc(-c2ccccc2)s1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.45
CTSL P07711 7/20 0.38
CTSS P25774 4/20 0.38
CTSB P07858 2/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
ALDH1A1 P00352 1/20 0.34
PAX8 Q06710 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043145 0.93 CTSK (0.49) CTSKCTSLCTSSCTSBMAPK1
SCHEMBL4048981 0.93 CTSK (0.43) CTSKCTSLCTSSCTSBCHRNB2
SCHEMBL4044586 0.92 CTSK (0.37) CTSKCTSSCHRNB2CHRNA7CHRNA4
SCHEMBL4044454 0.89 CTSK (0.55) CTSKCTSLCTSSCTSBCHRNB2
SCHEMBL4045083 0.89 CTSK (0.47) CTSKCTSLCTSSCTSBCHRNA7
SCHEMBL4050975 0.88 CTSK (0.43) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4038998 0.87 CTSK (0.44) CTSKCTSLCTSSCTSBCHRNA7
SCHEMBL4044003 0.87 CTSK (0.40) CTSKCTSLCTSSCTSBCHRNB2
SCHEMBL4048929 0.86 CTSK (0.52) CTSKCTSLCTSSCTSB
SCHEMBL4044220 0.86 CTSK (0.50) CTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed