SCHEMBL4048981

SCHEMBL4048981

CC(C)CC(NC(=O)Oc1ccc(-c2ccccn2)s1)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.43
CHRNB2 P17787 1/20 0.39
CHRNA7 P36544 1/20 0.39
CHRNA4 P43681 1/20 0.39
CTSL P07711 8/20 0.35
CTSS P25774 6/20 0.35
CTSB P07858 3/20 0.35
ALDH1A1 P00352 2/20 0.33
PAX8 Q06710 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042787 0.93 CHRNB2 (0.37) CTSKCHRNB2CHRNA7CHRNA4CTSS
SCHEMBL4045035 0.93 CTSK (0.45) CTSKCHRNB2CHRNA7CHRNA4CTSL
SCHEMBL4050975 0.86 CTSK (0.43) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4038998 0.85 CTSK (0.44) CTSKCHRNA7CTSLCTSSCTSB
SCHEMBL4045748 0.85 CTSK (0.51) CTSKCTSLCTSSCTSBALDH1A1
SCHEMBL4046924 0.85 CTSK (0.40) CTSKCHRNB2CHRNA7CHRNA4CTSL
SCHEMBL4043145 0.85 CTSK (0.49) CTSKCTSLCTSSCTSB
SCHEMBL4044586 0.85 CTSK (0.37) CTSKCHRNB2CHRNA7CHRNA4CTSS
SCHEMBL4042672 0.84 CTSK (0.41) CTSKCHRNB2CHRNA7CHRNA4CTSL
SCHEMBL4045083 0.84 CTSK (0.47) CTSKCHRNA7CTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed