SCHEMBL4044323

SCHEMBL4044323

O=C(NC(CC1CC1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1)Oc1cc2sccc2s1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.33
F2 P00734 1/20 0.33
GCK P35557 1/20 0.32
FKBP1A P62942 1/20 0.32
GPR132 Q9UNW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045303 0.92 CTSK (0.37) SMYD3FKBP1A
SCHEMBL4044199 0.92 SMYD3 (0.34) SMYD3F2FKBP1A
SCHEMBL4045954 0.91 SMYD3 (0.33) SMYD3FKBP1A
SCHEMBL4051011 0.90 HCRTR2 (0.34) SMYD3GCK
SCHEMBL6236087 0.90 SMYD3 (0.35) SMYD3F2GCKFKBP1AGPR132
SCHEMBL4044672 0.88 CTSV (0.33)
SCHEMBL4043092 0.88 CTSL (0.32) GCK
SCHEMBL4051435 0.87 HTRA1 (0.33) F2GPR132
SCHEMBL4048926 0.84 CTSL (0.39)
SCHEMBL4042904 0.83 CTSK (0.39) SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed