SCHEMBL4044199

SCHEMBL4044199

CCCC(NC(=O)Oc1cc2sccc2s1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.34
F2 P00734 6/20 0.32
F10 P00742 5/20 0.32
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP1A2 P05177 1/20 0.32
FKBP1A P62942 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045303 0.93 CTSK (0.37) SMYD3ALDH1A1FKBP1A
SCHEMBL4044323 0.92 SMYD3 (0.33) SMYD3F2FKBP1A
SCHEMBL4040719 0.91 SMYD3 (0.35) SMYD3CYP2C9CYP2C19ALDH1A1CYP1A2
SCHEMBL4043056 0.90 HSD17B10 (0.36) SMYD3TSHR
SCHEMBL4045954 0.90 SMYD3 (0.33) SMYD3ALDH1A1FKBP1ATSHR
SCHEMBL4050153 0.89 SMYD3 (0.35) SMYD3F2F10CYP2C9CYP2C19
SCHEMBL4042699 0.89 CTSK (0.32)
SCHEMBL4045509 0.88 PREP (0.33)
SCHEMBL4038641 0.88 CTSK (0.33) F2ALDH1A1
SCHEMBL4043393 0.86 FKBP1A (0.35) SMYD3FKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed