SCHEMBL4046215

SCHEMBL4046215

Cc1c(OC(=O)NC(Cc2cccs2)C(=O)N2CCC3C2C(=O)CN3S(=O)(=O)Cc2cccnc2)oc2ccccc12

nearest known ligand 0.34

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.34
CHRNA7 P36544 1/20 0.34
CHRNA4 P43681 1/20 0.34
GAA P10253 2/20 0.33
CTSB P07858 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33
SMYD3 Q9H7B4 2/20 0.32
USP2 O75604 3/20 0.32
LMNA P02545 3/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
NPSR1 Q6W5P4 3/20 0.32
TSHR P16473 2/20 0.32
HTT P42858 2/20 0.32
TP53 P04637 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
MAPT P10636 1/20 0.31
FKBP1A P62942 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050728 0.91 SMN1; SMN2 (0.33) CHRNB2CHRNA7CHRNA4GAACTSB
SCHEMBL4044165 0.90 CTSK (0.38) CHRNB2CHRNA7CHRNA4GAACTSB
SCHEMBL4049249 0.90 CHRNB2 (0.36) CHRNB2CHRNA7CHRNA4GAACTSS
SCHEMBL4048128 0.90 CHRNB2 (0.36) CHRNB2CHRNA7CHRNA4GAASMYD3
SCHEMBL4042344 0.89 CTSK (0.33) CHRNB2CHRNA7CHRNA4GAACTSK
SCHEMBL4045248 0.89 NPC1 (0.33) GAACTSBCTSSCTSKLMNA
SCHEMBL4044961 0.89 CHRNB2 (0.35) CHRNB2CHRNA7CHRNA4GAACTSB
SCHEMBL4047038 0.86 CTSK (0.39) CTSBCTSSCTSK
SCHEMBL4046790 0.84 USP30 (0.36) CTSBCTSSCTSK
SCHEMBL4045954 0.83 SMYD3 (0.33) CHRNA7CTSBCTSSCTSKSMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed