SCHEMBL4050728

SCHEMBL4050728

Cc1c(OC(=O)NC(Cc2cccs2)C(=O)N2CCC3C2C(=O)CN3S(=O)(=O)c2cccnc2)oc2ccccc12

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.33
USP2 O75604 3/20 0.33
LMNA P02545 3/20 0.33
NPSR1 Q6W5P4 3/20 0.33
GAA P10253 2/20 0.33
TSHR P16473 2/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNA7 P36544 1/20 0.33
CHRNA4 P43681 1/20 0.33
HTT P42858 2/20 0.32
TP53 P04637 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
HSD17B10 Q99714 1/20 0.32
KCNQ1 P51787 1/20 0.32
CTSK P43235 3/20 0.31
POLB P06746 1/20 0.31
GBA1 P04062 1/20 0.30
CTSB P07858 1/20 0.30
CTSS P25774 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046215 0.91 CHRNB2 (0.34) SMN1; SMN2USP2LMNANPSR1GAA
SCHEMBL4042344 0.91 CTSK (0.33) SMN1; SMN2GAACHRNB2CHRNA7CHRNA4
SCHEMBL4039790 0.90 CTSK (0.39) SMN1; SMN2USP2LMNANPSR1GAA
SCHEMBL4046064 0.89 SMN1; SMN2 (0.35) SMN1; SMN2USP2LMNAGAACTSK
SCHEMBL4042714 0.89 SMN1; SMN2 (0.36) SMN1; SMN2USP2LMNANPSR1GAA
SCHEMBL4047038 0.89 CTSK (0.39) CTSKCTSBCTSS
SCHEMBL4044961 0.86 CHRNB2 (0.35) SMN1; SMN2USP2LMNANPSR1GAA
SCHEMBL4046790 0.86 USP30 (0.36) CTSKCTSBCTSS
SCHEMBL4045248 0.86 NPC1 (0.33) SMN1; SMN2LMNAGAATSHRCTSK
SCHEMBL4045719 0.85 SMN1; SMN2 (0.32) SMN1; SMN2CTSKCTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed