SCHEMBL404720

SCHEMBL404720

CCCCCCOc1c(CC)cccc1C(Oc1cnnnc1-c1ccccc1)c1cccc(CC)c1OCCCCCC

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SOAT1 P35610 1/20 0.39
CYSLTR2 Q9NS75 2/20 0.34
CYSLTR1 Q9Y271 2/20 0.34
PTPN1 P18031 1/20 0.33
PTPN11 Q06124 1/20 0.32
PPARG P37231 3/20 0.32
PTGES O14684 1/20 0.32
ALOX5 P09917 1/20 0.32
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
PIK3CD O00329 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2018229 0.82 SOAT1 (0.41) SOAT1PTPN11PPARG
SCHEMBL1984480 0.80 SOAT1 (0.41) SOAT1ALOX5
SCHEMBL118832 0.80 SOAT1 (0.41) SOAT1ALOX5
SCHEMBL28980883 0.76 SOAT1 (0.42) SOAT1PTPN11PPARGMEN1CYP1A2
SCHEMBL29189935 0.76 SOAT1 (0.40) SOAT1PTPN11PPARGALOX5MEN1
SCHEMBL1276212 0.75 SOAT1 (0.40) SOAT1PTPN11ALOX5MEN1CYP1A2
Phenol SCHEMBL28102520 0.73 L3MBTL1 (0.40) SOAT1PPARGALOX5MEN1CYP3A4
SCHEMBL25315299 0.73
SCHEMBL28296116 0.73 SOAT1 (0.40) SOAT1ALOX5
SCHEMBL64304 0.73 SOAT1 (0.40) SOAT1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 257 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024126253-A1 COMPOSITION COMPRISING A UV-SCREENING AGENT, A SUITABLY SELECTED LIPOPHILIC POLYMER AND A CARRAGEENAN L'OREAL (FR) 2024-06-20 WO claimed
WO-2024106520-A1 NON-STICKY STABLE COMPOSITION WITH TEXTURE TRANSFORMATION PROPERTY L'OREAL (FR) 2024-05-23 WO claimed
EP-3393437-B1 PHOTOPROTECTIVE COMPOSITION BASED ON A CARBOXYLIC ACID ESTER; USE OF SAID COMPOUND FOR INCREASING THE SUN PROTECTION FACTOR OREAL (FR) 2023-06-07 EP claimed
US-10918583-B2 Cosmetic or dermatological composition comprising a merocyanine, an organic UVB-screening agent and an additional organic UVA-screening agent L'OREAL (FR) 2021-02-16 US claimed
EP-3193816-B1 COMPOSITION BASED ON MULTILAYER SPHERICAL COMPOSITE PARTICLES AND ON A UV-SCREENING AGENT OREAL (FR) 2020-05-13 EP claimed
US-20190336421-A1 COMPOSITION COMPRISING RESORCINOL OR DERIVATIVE THEREOF L'OREAL (FR) 2019-11-07 US claimed
EP-2775994-B1 COMPOSITION WITH A CONTINUOUS OIL PHASE CONTAINING AT LEAST ONE LIPOPHILIC ORGANIC UV-SCREENING AGENT AND HYDROPHOBIC SILICA AEROGEL PARTICLES OREAL (FR) 2019-10-16 EP claimed
EP-3016631-B1 COSMETIC COMPOSITION OREAL (FR) 2019-10-02 EP claimed
US-10272021-B2 Composition based on multilayer spherical composite particles and on a UV-screening agent L'OREAL (FR) 2019-04-30 US claimed
US-20180369094-A1 PHOTOPROTECTIVE COMPOSITION BASED ON A CARBOXYLIC ACID ESTER; USE OF SAID COMPOUND FOR INCREASING THE SUN PROTECTION FACTOR L'OREAL (FR) 2018-12-27 US claimed
WO-2013084184-A2 PHOTOPROTECTIVE AND SELF-TANNING COSMETIC EMULSIONS L'OREAL (FR) 2013-06-13 WO claimed
WO-2013068237-A1 COMPOSITION WITH A CONTINUOUS OIL PHASE CONTAINING AT LEAST ONE LIPOPHILIC ORGANIC UV-SCREENING AGENT AND HYDROPHOBIC SILICA AEROGEL PARTICLES L'OREAL (FR) 2013-05-16 WO claimed
US-20130058990-A1 COMPOSITION CONTAINING A DIBENZOYLMETHANE SCREENING AGENT AND A HYDROPHILIC OR WATER-SOLUBLE MEROCYANIN UV-SCREENING AGENT; PROCESS FOR PHOTOSTABILIZING THE DIBENZOYLMETHANE SCREENING AGENT L'OREAL (FR) 2013-03-07 US claimed
EP-2547313-A1 COMPOSITION CONTAINING A DIBENZOYLMETHANE SCREENING AGENT AND A HYDROPHILIC OR WATER-SOLUBLE MEROCYANIN UV-SCREENING AGENT; PROCESS FOR PHOTOSTABILIZING THE DIBENZOYLMETHANE SCREENING AGENT L'Oréal (FR) 2013-01-23 EP claimed
WO-2012168102-A2 ANHYDROUS ANTISUN CREAM COMPRISING A NON-EMULSIFYING ELASTOMERIC ORGANOPOLYSILOXANE, A MATTING AGENT AND A NON-SILICONE ORGANIC OIL THICKENER L'OREAL (FR) 2012-12-13 WO claimed
EP-2174644-B1 Cosmetic composition comprising a dibenzoylmethane derivative and a dithiolane; Photostabilization of a dibenzoylmethane derivative OREAL (FR) 2012-11-14 EP claimed
WO-2011113718-A1 COMPOSITION CONTAINING A DIBENZOYLMETHANE SCREENING AGENT AND A HYDROPHILIC OR WATER-SOLUBLE MEROCYANIN UV-SCREENING AGENT; PROCESS FOR PHOTOSTABILIZING THE DIBENZOYLMETHANE SCREENING AGENT L'OREAL (FR) 2011-09-22 WO claimed
US-20100172944-A1 COMBINATION OF MONOSACCHARIDES WITH SUNSCREENS AND USE THEREOF L'OREAL (FR) 2010-07-08 US claimed
US-20100086502-A1 Cosmetic/sunscreen compositions containing dibenzoylmethane compounds and dithiolane compound photostabilizers therefor L'OREAL (FR) 2010-04-08 US claimed
US-20090285868-A1 Photostable cosmetic compositions comprising dibenzoylmethane/pyrrolidinone compounds L'OREAL (FR) 2009-11-19 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190336421-A1 COMPOSITION COMPRISING RESORCINOL OR DERIVATIVE THEREOF NQO1, LRAT, RBP4 SOAT1 489/4885CYSLTR2 3186/4885CYSLTR1 3206/4885
US-20100086502-A1 Cosmetic/sunscreen compositions containing dibenzoylmethane compounds and dithiolane compound photostabilizers therefor NOTUM, DDT, FDFT1 SOAT1 20/4885CYSLTR2 2091/4885CYSLTR1 1885/4885
US-20090285868-A1 Photostable cosmetic compositions comprising dibenzoylmethane/pyrrolidinone compounds NOTUM, CYP51A1, DHPS SOAT1 81/4885CYSLTR2 2521/4885CYSLTR1 2371/4885
US-10272021-B2 Composition based on multilayer spherical composite particles and on a UV-screening agent CUTA, RAD52, PSMC3 SOAT1 3955/4885CYSLTR2 3504/4885CYSLTR1 3424/4885
US-20130058990-A1 COMPOSITION CONTAINING A DIBENZOYLMETHANE SCREENING AGENT AND A HYDROPHILIC OR WATER-SOLUBLE MEROCYANIN UV-SCREENING AGENT; PROCESS FOR PHOTOSTABILIZING THE DIBENZOYLMETHANE SCREENING AGENT CRYZ, MSH6, TYR SOAT1 1427/4885CYSLTR2 2100/4885CYSLTR1 2482/4885
US-10918583-B2 Cosmetic or dermatological composition comprising a merocyanine, an organic UVB-screening agent and an additional organic UVA-screening agent KRT18, CRYZ, CUTA SOAT1 2475/4885CYSLTR2 1175/4885CYSLTR1 2202/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.