SCHEMBL4047237

SCHEMBL4047237

CC(C)(C)CC(NC(=O)Oc1ccsc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.35
CTSK P43235 2/20 0.34
FKBP1A P62942 1/20 0.33
CTSL P07711 1/20 0.32
CTSS P25774 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045208 0.93 SMYD3 (0.35) SMYD3FKBP1AALDH1A1CYP2C9TSHR
SCHEMBL4042764 0.93 CTSK (0.38) SMYD3CTSKFKBP1ACTSLCTSS
SCHEMBL4046102 0.90 KCNQ1 (0.38) SMYD3CTSKALDH1A1TSHR
SCHEMBL4045926 0.89 GPR132 (0.36) FKBP1ACTSLCTSS
SCHEMBL4045044 0.88 CTSK (0.36) CTSK
SCHEMBL4049268 0.88 SMYD3 (0.35) SMYD3CTSKFKBP1ACTSLCTSS
SCHEMBL4045469 0.87 ELANE (0.37) CTSKCTSLCTSSALDH1A1
SCHEMBL4048509 0.87 CTSK (0.38) CTSKALDH1A1
SCHEMBL4045645 0.86 SMYD3 (0.34) SMYD3CTSKFKBP1ACTSLCTSS
SCHEMBL4051200 0.83 CTSK (0.44) CTSKCTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed