SCHEMBL4048544

SCHEMBL4048544

CCCC(NC(=O)Oc1ccoc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccc[n+]([O-])c1

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
P2RY12 Q9H244 1/20 0.32
CTSK P43235 2/20 0.32
PREP P48147 1/20 0.30
FAP Q12884 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4040755 0.93 CTSK (0.35) CTSK
SCHEMBL4047629 0.92 CTSK (0.40) CTSK
SCHEMBL4042622 0.89 CTSS (0.40) CTSK
SCHEMBL4044695 0.89 CTSK (0.36) P2RY12CTSK
SCHEMBL4044073 0.89 CTSK (0.33) CTSKPREPFAP
SCHEMBL4044048 0.88 HSD17B10 (0.37) CTSKPREPFAP
SCHEMBL4046811 0.88 CTSK (0.33) P2RY12CTSKPREPFAP
SCHEMBL4047785 0.87 CTSK (0.32) CTSKPREPFAP
SCHEMBL4045249 0.87 CTSK (0.36) P2RY12CTSK
SCHEMBL4048294 0.86 ALDH1A1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed