SCHEMBL4048878

SCHEMBL4048878

CCSNCCCCC(NC(=O)O)c1c[nH]c(-c2ccccc2)n1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 9/20 0.33
HDAC6 Q9UBN7 8/20 0.33
HDAC3 O15379 8/20 0.33
HDAC2 Q92769 8/20 0.33
HDAC8 Q9BY41 8/20 0.33
HDAC4 P56524 4/20 0.33
HDAC7 Q8WUI4 4/20 0.33
HDAC10 Q969S8 4/20 0.33
HDAC11 Q96DB2 4/20 0.33
HDAC9 Q9UKV0 4/20 0.33
HDAC5 Q9UQL6 4/20 0.33
ADORA3 P0DMS8 2/20 0.33
ADORA2A P29274 2/20 0.33
ADORA1 P30542 1/20 0.33
TACR3 P29371 3/20 0.33
PDE2A O00408 2/20 0.32
ALDH1A1 P00352 1/20 0.31
PIN1 Q13526 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3955607 0.82 SIRT1 (0.42) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL4048868 0.82 ADORA3 (0.41) HDAC1HDAC6ADORA3ADORA2AADORA1
SCHEMBL5469798 0.80 HDAC6 (0.52) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL4052446 0.79 MAPT (0.47) ALDH1A1
SCHEMBL4048617 0.77 KDM4E (0.43) ALDH1A1
SCHEMBL4048438 0.76 HDAC1 (0.52) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL5461533 0.75 HDAC6 (0.44) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL393077 0.74 F11 (0.40) TACR3ALDH1A1
SCHEMBL5355871 0.72 HDAC1 (0.39) HDAC1HDAC6ADORA3ADORA2APDE2A
SCHEMBL5363436 0.72 HDAC6 (0.55) HDAC1HDAC6HDAC3HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026701-A1 SIRTUIN INHIBITORS METHYLGENE INC. (CA) 2009-03-05 WO disclosed