SCHEMBL4049526

SCHEMBL4049526

CNC(=S)NCCCCC(NC(=O)O)c1n[nH]c(-c2ccccc2)n1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 10/20 0.38
ADORA2A P29274 9/20 0.38
ADORA1 P30542 6/20 0.36
HRH2 P25021 2/20 0.35
HRH4 Q9H3N8 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
F2 P00734 1/20 0.34
F12 P00748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050458 0.88 CYP1A2 (0.41) ADORA3ADORA2AADORA1TP53CYP1A2
SCHEMBL4047830 0.82 MAPT (0.47)
SCHEMBL4048868 0.81 ADORA3 (0.41) ADORA3ADORA2AADORA1TP53CYP1A2
SCHEMBL4051945 0.81 CYP1A2 (0.43) ADORA3ADORA2AADORA1CYP1A2F2
SCHEMBL5360457 0.80 HDAC6 (0.53) HDAC1HDAC6
SCHEMBL4052271 0.76 HDAC3 (0.41) HDAC1HDAC6
SCHEMBL4050469 0.75 CYP1A2 (0.40) ADORA3ADORA2AADORA1CYP1A2HDAC1
SCHEMBL3959226 0.75 ALDH1A1 (0.56) CYP1A2HDAC1HDAC6
SCHEMBL5363015 0.72 MAPT (0.60) HDAC1HDAC6
SCHEMBL3955607 0.71 SIRT1 (0.42) ADORA3HDAC1HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009026701-A1 SIRTUIN INHIBITORS METHYLGENE INC. (CA) 2009-03-05 WO disclosed