SCHEMBL4049555

SCHEMBL4049555

COc1ccc2oc(OC(=O)NC3(C(=O)N4CCC5C4C(=O)CN5C(=O)Cc4cccnc4)CCCCC3)cc2c1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.41
CHRNA7 P36544 1/20 0.41
CHRNA4 P43681 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HPGD P15428 1/20 0.40
IDO1 P14902 1/20 0.36
TACR2 P21452 1/20 0.35
MAPT P10636 2/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
C3AR1 Q16581 1/20 0.34
KMT2A Q03164 1/20 0.34
POLB P06746 1/20 0.33
TP53 P04637 1/20 0.33
NAMPT P43490 2/20 0.33
KLK7 P49862 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043466 0.88 CHRNB2 (0.40) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4045182 0.85 KCNQ1 (0.37) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4046100 0.84 KLK7 (0.35) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4047235 0.83 CTSL (0.36) ALDH1A1HPGDTACR2KDM4EGAA
SCHEMBL4047073 0.83 CHRNB2 (0.43) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4043880 0.82 CHRNB2 (0.41) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4044034 0.82 CHRNB2 (0.41) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4041874 0.81 CHRNB2 (0.37) CHRNB2CHRNA7CHRNA4MAPTGAA
SCHEMBL4044847 0.80 CHRNB2 (0.39) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4050955 0.80 CTSK (0.37) HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed