SCHEMBL4048186

SCHEMBL4048186

CCCC(NC(=O)Oc1ccc2ncccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccc[n+]1[O-]

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
PREP P48147 2/20 0.34
FAP Q12884 2/20 0.34
RAB9A P51151 3/20 0.32
CTSK P43235 3/20 0.32
NR2F2 P24468 2/20 0.32
PPARG P37231 2/20 0.32
PPARA Q07869 1/20 0.32
MAPT P10636 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KDM4E B2RXH2 1/20 0.31
TNF P01375 1/20 0.31
LMNA P02545 1/20 0.31
NOD1 Q9Y239 1/20 0.31
ALOX5 P09917 1/20 0.31
CHRM5 P08912 1/20 0.31
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31
P2RY12 Q9H244 1/20 0.30
EPHX2 P34913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047523 0.93 CTSK (0.39) ALDH1A1CTSK
SCHEMBL4049558 0.92 CTSK (0.36) CTSK
SCHEMBL4043292 0.90 ALDH1A1 (0.37) ALDH1A1PREPFAPRAB9ACTSK
SCHEMBL4046799 0.88 ALDH1A1 (0.39) ALDH1A1PREPFAPCTSK
SCHEMBL4041133 0.87 CTSK (0.36) ALDH1A1PREPFAPCTSKP2RY12
SCHEMBL4046989 0.86 ALDH1A1 (0.38) ALDH1A1PREPFAPRAB9ANR2F2
SCHEMBL4039771 0.85 ALDH1A1 (0.38) ALDH1A1PREPFAPRAB9ACTSK
SCHEMBL4043678 0.85 ALDH1A1 (0.38) ALDH1A1PREPFAPRAB9ACTSK
SCHEMBL4050306 0.85 PKM (0.36) ALDH1A1CTSKKDM4ELMNACHRM5
SCHEMBL4045359 0.85 PREP (0.33) PREPFAPCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed