SCHEMBL4051337

SCHEMBL4051337

COc1cccc2cc(OC(=O)NC(CC(C)C)C(=O)N3CCC4C3C(=O)CN4C(=O)Cc3cccnc3)oc12

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.43
CHRNA7 P36544 3/20 0.43
CHRNA4 P43681 3/20 0.43
CTSK P43235 2/20 0.39
IDO1 P14902 2/20 0.35
ALDH1A1 P00352 2/20 0.35
PAX8 Q06710 1/20 0.35
USP2 O75604 1/20 0.35
MAPT P10636 1/20 0.35
PPARG P37231 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
TSHR P16473 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
MMP1 P03956 1/20 0.33
MMP3 P08254 1/20 0.33
MMP9 P14780 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046927 0.93 CHRNA7 (0.41) CHRNB2CHRNA7CHRNA4CTSKIDO1
SCHEMBL4042383 0.89 CTSK (0.42) CHRNB2CHRNA7CHRNA4CTSKMMP1
SCHEMBL4043180 0.88 CHRNB2 (0.42) CHRNB2CHRNA7CHRNA4CTSKALDH1A1
SCHEMBL4047073 0.87 CHRNB2 (0.43) CHRNB2CHRNA7CHRNA4CTSKIDO1
SCHEMBL4044616 0.86 CHRNB2 (0.39) CHRNB2CHRNA7CHRNA4CTSKALDH1A1
SCHEMBL4043435 0.84 CTSK (0.38) CHRNB2CHRNA7CHRNA4CTSKALDH1A1
SCHEMBL4044450 0.84 CTSK (0.43) CTSKALDH1A1PAX8
SCHEMBL4040201 0.84 CTSK (0.45) CTSKALDH1A1NPSR1
SCHEMBL4045179 0.83 CTSK (0.44) CHRNA7CTSKPAX8MMP1MMP3
SCHEMBL4050975 0.82 CTSK (0.43) CTSKALDH1A1PAX8MMP1MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed