SCHEMBL4043435

SCHEMBL4043435

COc1cccc2cc(OC(=O)NC(CC(C)C)C(=O)N3CCC4C3C(=O)CN4S(=O)(=O)C(=O)c3cccnc3)oc12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.38
CHRNB2 P17787 3/20 0.38
CHRNA7 P36544 3/20 0.38
CHRNA4 P43681 3/20 0.38
AAK1 Q2M2I8 1/20 0.34
MMP1 P03956 1/20 0.33
MMP3 P08254 1/20 0.33
MMP9 P14780 1/20 0.33
ALDH1A1 P00352 3/20 0.33
KDM4E B2RXH2 3/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
USP2 O75604 1/20 0.32
PPARG P37231 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PREP P48147 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4039150 0.93 CHRNA7 (0.36) CTSKCHRNB2CHRNA7CHRNA4ALDH1A1
SCHEMBL4044616 0.91 CHRNB2 (0.39) CTSKCHRNB2CHRNA7CHRNA4MMP1
SCHEMBL4045633 0.89 CTSK (0.41) CTSKMMP1MMP3MMP9ALDH1A1
SCHEMBL4043180 0.89 CHRNB2 (0.42) CTSKCHRNB2CHRNA7CHRNA4ALDH1A1
SCHEMBL4049357 0.88 CTSK (0.37) CTSKALDH1A1KDM4ERAB9AHPGD
SCHEMBL4049366 0.88 CTSK (0.38) CTSKCHRNB2CHRNA7CHRNA4AAK1
SCHEMBL4045839 0.85 CTSK (0.45) CTSK
SCHEMBL4047069 0.85 CTSK (0.42) CTSKMMP1MMP3MMP9PREP
SCHEMBL4051337 0.84 CHRNB2 (0.43) CTSKCHRNB2CHRNA7CHRNA4MMP1
SCHEMBL4043183 0.84 CTSK (0.43) CTSKMMP1MMP3MMP9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed