SCHEMBL4044616

SCHEMBL4044616

COc1cccc2cc(OC(=O)NC(CC(C)C)C(=O)N3CCC4C3C(=O)CN4S(=O)(=O)c3cccnc3)oc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.39
CHRNA7 P36544 3/20 0.39
CHRNA4 P43681 3/20 0.39
CTSK P43235 6/20 0.36
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
PPARG P37231 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RXFP1 Q9HBX9 1/20 0.35
NCOR2 Q9Y618 1/20 0.35
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
NPC1 O15118 1/20 0.34
KCNQ1 P51787 1/20 0.33
HCRTR2 O43614 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA2B P29275 1/20 0.33
ADORA1 P30542 1/20 0.33
CTSL P07711 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042524 0.93 CHRNA7 (0.37) CHRNB2CHRNA7CHRNA4USP2ALDH1A1
SCHEMBL4043180 0.91 CHRNB2 (0.42) CHRNB2CHRNA7CHRNA4CTSKUSP2
SCHEMBL4043435 0.91 CTSK (0.38) CHRNB2CHRNA7CHRNA4CTSKUSP2
SCHEMBL4050961 0.89 CTSK (0.36) CHRNA7CTSKALDH1A1RXFP1HSD17B10
SCHEMBL4043843 0.89 CTSK (0.41) CTSKHSD17B10HCRTR2CTSLCTSS
SCHEMBL4045839 0.88 CTSK (0.45) CTSKCTSLCTSSCTSVCTSB
SCHEMBL4047148 0.87 CHRNB2 (0.39) CHRNB2CHRNA7CHRNA4CTSKALDH1A1
SCHEMBL4051337 0.86 CHRNB2 (0.43) CHRNB2CHRNA7CHRNA4CTSKUSP2
SCHEMBL4043661 0.85 ALDH1A1 (0.38) CTSKALDH1A1NPC1CTSLCTSS
SCHEMBL4049357 0.85 CTSK (0.37) CTSKALDH1A1NPC1CTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed