SCHEMBL4043180

SCHEMBL4043180

COc1cccc2cc(OC(=O)NC(CC(C)C)C(=O)N3CCC4C3C(=O)CN4S(=O)(=O)Cc3cccnc3)oc12

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.42
CHRNA7 P36544 3/20 0.42
CHRNA4 P43681 3/20 0.42
CTSK P43235 2/20 0.35
SMYD3 Q9H7B4 2/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
PPARG P37231 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
NCOR2 Q9Y618 1/20 0.34
NPC1 O15118 2/20 0.33
KMT2A Q03164 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
TSHR P16473 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043632 0.93 CHRNA7 (0.40) CHRNB2CHRNA7CHRNA4SMYD3USP2
SCHEMBL4044616 0.91 CHRNB2 (0.39) CHRNB2CHRNA7CHRNA4CTSKUSP2
SCHEMBL4040754 0.89 CTSK (0.40) CHRNB2CHRNA7CHRNA4CTSK
SCHEMBL4043435 0.89 CTSK (0.38) CHRNB2CHRNA7CHRNA4CTSKUSP2
SCHEMBL4043661 0.88 ALDH1A1 (0.38) CTSKALDH1A1NPC1
SCHEMBL4051337 0.88 CHRNB2 (0.43) CHRNB2CHRNA7CHRNA4CTSKUSP2
SCHEMBL4046703 0.88 CHRNB2 (0.42) CHRNB2CHRNA7CHRNA4CTSKSMYD3
SCHEMBL4045839 0.85 CTSK (0.45) CTSK
SCHEMBL4044807 0.85 CTSK (0.39) CTSKSMYD3ALDH1A1
SCHEMBL4050147 0.84 CTSK (0.40) CTSKSMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed
WO-2009024766-A2 DYEING PROCESS IN IONIC LIQUID SOLVENTS THE QUEEN'S UNIVERSITY OF BELFAST (GB) 2009-02-26 WO disclosed
US-4359322-A FOR FIBER-REACTIVE DYES ON CELLULOSE NEAL CHEMICAL COMPANY, INC. (US) 1982-11-16 US disclosed