SCHEMBL4055359

SCHEMBL4055359

O=[N+]([O-])c1ccc(Cl)c(-c2ncc[nH]2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.49
CCNB2 O95067 1/20 0.47
CDK1 P06493 1/20 0.47
CCNB1 P14635 1/20 0.47
CCNA2 P20248 1/20 0.47
CDK2 P24941 1/20 0.47
CCNA1 P78396 1/20 0.47
CCNB3 Q8WWL7 1/20 0.47
NPBWR1 P48145 5/20 0.47
GSK3B P49841 1/20 0.46
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
HSP90AA1 P07900 1/20 0.44
AGTR1 P30556 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 1/20 0.44
TDP1 Q9NUW8 2/20 0.44
CYP3A4 P08684 2/20 0.44
PTPRC P08575 1/20 0.44
S100A4 P26447 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5747525 0.84 MEN1 (0.46) NPBWR1MEN1NPC1HSP90AA1AGTR1
SCHEMBL9292469 0.82 NPC1 (0.44) NPBWR1GSK3BMEN1NPC1HSP90AA1
SCHEMBL8539529 0.82 GPR35 (0.49) NPBWR1MEN1NPC1HSP90AA1AGTR1
SCHEMBL5249670 0.82 MAPT (0.56) GSK3BMEN1NPC1HSP90AA1AGTR1
SCHEMBL8540776 0.81 AMY1A (0.48) NPBWR1GSK3BMEN1NPC1HSP90AA1
SCHEMBL31463535 0.81 AMY1A (0.48) NPBWR1GSK3BMEN1NPC1HSP90AA1
SCHEMBL8615132 0.79 NPC1 (0.42) NPBWR1GSK3BMEN1NPC1HSP90AA1
SCHEMBL10440889 0.79 ABCC8 (0.43) GSK3BMEN1NPC1HSP90AA1AGTR1
SCHEMBL8536767 0.79 CYP3A4 (0.46) NPBWR1MEN1NPC1HSP90AA1AGTR1
SCHEMBL8536769 0.79 NPC1 (0.42) NPBWR1GSK3BMEN1NPC1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009030952-A2 PHENYLCARBOXAMIDE DERIVATIVES AS INHIBITORS AND EFFECTORS OF THE HEDGEHOG PATHWAY ASTRAZENECA AB (SE) 2009-03-12 WO disclosed