SCHEMBL8536767

SCHEMBL8536767

O=[N+]([O-])c1ccc(C=S)c(-c2ncc[nH]2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.46
NAMPT P43490 1/20 0.46
XDH P47989 1/20 0.46
NPC1 O15118 5/20 0.42
RAB9A P51151 5/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
PARP1 P09874 1/20 0.42
HSP90AA1 P07900 1/20 0.42
AGTR1 P30556 1/20 0.42
MAPT P10636 5/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
KDM4E B2RXH2 1/20 0.41
METAP1 P53582 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PKN1 Q16512 1/20 0.41
PKN2 Q16513 1/20 0.41
TDP1 Q9NUW8 3/20 0.41
HTT P42858 2/20 0.41
MMP2 P08253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5747525 0.83 MEN1 (0.46) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL8539360 0.81 ERN1 (0.49) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL4055359 0.79 HSD17B10 (0.49) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL9292469 0.79 NPC1 (0.44) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL8539529 0.79 GPR35 (0.49) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL5249670 0.79 MAPT (0.56) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL31463535 0.77 AMY1A (0.48) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL8540776 0.77 AMY1A (0.48) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL8615132 0.76 NPC1 (0.42) CYP3A4NAMPTXDHNPC1RAB9A
SCHEMBL10440889 0.76 ABCC8 (0.43) CYP3A4NAMPTXDHNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed