SCHEMBL8540776

SCHEMBL8540776

O=[N+]([O-])c1ccc(-c2ncc[nH]2)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 2/20 0.48
NPC1 O15118 4/20 0.46
RAB9A P51151 3/20 0.46
MEN1 O00255 1/20 0.46
HSP90AA1 P07900 1/20 0.46
AGTR1 P30556 1/20 0.46
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 2/20 0.44
HIF1A Q16665 1/20 0.44
CYP3A4 P08684 2/20 0.43
NAMPT P43490 1/20 0.43
XDH P47989 1/20 0.43
TDP1 Q9NUW8 2/20 0.41
PTPRC P08575 1/20 0.41
S100A4 P26447 1/20 0.41
MAPT P10636 4/20 0.40
GSK3B P49841 1/20 0.40
KDM4E B2RXH2 1/20 0.39
METAP1 P53582 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31463535 1.00 AMY1A (0.48) AMY1ANPC1RAB9AMEN1HSP90AA1
SCHEMBL8539529 0.83 GPR35 (0.49) NPC1RAB9AMEN1HSP90AA1AGTR1
SCHEMBL5249670 0.83 MAPT (0.56) NPC1RAB9AMEN1HSP90AA1AGTR1
SCHEMBL5747525 0.82 MEN1 (0.46) NPC1RAB9AMEN1HSP90AA1AGTR1
SCHEMBL9292469 0.81 NPC1 (0.44) NPC1RAB9AMEN1HSP90AA1AGTR1
SCHEMBL4055359 0.81 HSD17B10 (0.49) NPC1RAB9AMEN1HSP90AA1AGTR1
SCHEMBL10440889 0.80 ABCC8 (0.43) NPC1RAB9AMEN1HSP90AA1AGTR1
SCHEMBL8536769 0.80 NPC1 (0.42) NPC1RAB9AMEN1HSP90AA1AGTR1
SCHEMBL8539360 0.79 ERN1 (0.49) NPC1RAB9AMEN1HSP90AA1AGTR1
SCHEMBL8536108 0.78 HTT (0.51) AMY1ANPC1RAB9AMEN1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0857171-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1998-08-12 EP disclosed
WO-1997031917-A9 SUBSTITUTED PHENYLOXAZOLIDINONES AND THEIR USE AS ANTIBIOTICS 1997-10-30 WO disclosed
WO-1997015555-A2 IMIDAZOLE DERIVATIVES AND THE USE THEREOF AS NITROGEN MONOXIDE SYNTHASE INHIBITORS SCHERING AKTIENGESELLSCHAFT (DE) 1997-05-01 WO disclosed