SCHEMBL4059533

SCHEMBL4059533

O=C(OCCc1ccccc1)n1ccnc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 1/20 0.48
GRIN2B Q13224 1/20 0.46
HCAR2 Q8TDS4 1/20 0.44
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
ALDH1A1 P00352 1/20 0.42
TP53 P04637 1/20 0.42
GLA P06280 1/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HIF1A Q16665 1/20 0.42
HSD17B10 Q99714 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
AKR1B10 O60218 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23764025 0.92 LMNA (0.51) NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL6095146 0.90 CYP3A4 (0.42) P2RX4GRIN2BALDH1A1CYP3A4
SCHEMBL20635282 0.87 CYP2D6 (0.46) TDP1CYP3A4
SCHEMBL432657 0.85 KMT2A (0.49) P2RX4GRIN2BTDP1NPC1RAB9A
SCHEMBL26597537 0.84 TBXAS1 (0.52) NPC1RAB9AALDH1A1CYP3A4HPGD
SCHEMBL15435863 0.84 CYP19A1 (0.49) FAAHMGLL
SCHEMBL12016623 0.84 ALDH1A1 (0.39) TDP1ALDH1A1
SCHEMBL6101374 0.84 QPCT (0.42) HCAR2CYP3A4FAAHMGLL
SCHEMBL19973625 0.83 CA12 (0.50) NPC1RAB9AALDH1A1CYP3A4SMN1; SMN2
SCHEMBL12964049 0.82 FAAH (0.45) ALDH1A1CYP3A4HPGDTSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114787139-B Methods and intermediates for preparing MCL1 inhibitors 吉利德科学公司 2025-03-11 CN disclosed
CN-114787139-A Processes and intermediates for preparing MCL1 inhibitors 吉利德科学公司 2022-07-22 CN disclosed
EP-2012759-A1 PURINE DERIVATIVES AS A2A RECEPTOR AGONISTS Novartis AG (CH) 2009-01-14 EP disclosed
WO-2007121923-A1 PURINE DERIVATIVES AS A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2007-11-01 WO disclosed
US-20060094880-A9 Synthetic process for trans-aminocyclohexyl ether compounds BARRETT ANTHONY G M 2006-05-04 US disclosed
US-20050038256-A1 Synthetic process for trans-aminocyclohexyl ether compounds CARDIOME PHARMA CORP. (CA) 2005-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060094880-A9 Synthetic process for trans-aminocyclohexyl ether compounds AKR1C3, CBR1, CBR3 P2RX4 4721/4885GRIN2B 2196/4885HCAR2 185/4885
US-20050038256-A1 Synthetic process for trans-aminocyclohexyl ether compounds AKR1C3, CBR1, CBR3 P2RX4 4721/4885GRIN2B 2196/4885HCAR2 185/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.